Phenibut (hydrochloride)

CAS No. 3060-41-1

Phenibut (hydrochloride)( 3-Amino-4-phenylbutyric acid hydrochloride )

Catalog No. M22204 CAS No. 3060-41-1

Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates dopamine receptors, and inhibits the actions of β-phenethylamine.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
100MG 53 In Stock
200MG 84 In Stock
500MG 159 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Phenibut (hydrochloride)
  • Note
    Research use only, not for human use.
  • Brief Description
    Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates dopamine receptors, and inhibits the actions of β-phenethylamine.
  • Description
    Phenibut (hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors, blocks α2δ subunit-containing voltage-gated calcium channels, stimulates dopamine receptors, and inhibits the actions of β-phenethylamine.
  • In Vitro
    Phenibut hydrochloride is a neuropsychotropic agent. Phenibut hydrochloride also stimulates dopamine receptors and antagonizes β-phenethylamine (PEA), a putative endogenous anxiogenic.
  • In Vivo
    ——
  • Synonyms
    3-Amino-4-phenylbutyric acid hydrochloride
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GABAB
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    3060-41-1
  • Formula Weight
    215.68
  • Molecular Formula
    C10H14ClNO2
  • Purity
    >98% (HPLC)
  • Solubility
    In Vitro:?H2O : 100 mg/mL (463.65 mM)
  • SMILES
    NC[C@@]([H])(CC(=O)O)c1ccccc1.[Cl]
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Zvejniece L , Vavers E , Svalbe B , et al. R-phenibut binds to the α2-δ subunit of voltage-dependent calcium channels and exerts gabapentin-like anti-nociceptive effects.[J]. Pharmacol Biochem Behav, 2015:23-29.
molnova catalog
related products
  • NPR-C activator 1

    NPR-C activator 1 (Compound 1) is a potent agonist (EC50 ~ 1 μM) of natriuretic peptide receptor C (NPR-C), which plays a crucial role in regulating vascular homeostasis, and demonstrates promising in vivo pharmacokinetic properties .

  • Phellodendrine

    Phellodendrine has anti-nephritic activity, may be due to its ability to inhibit the proliferation or the migration of macrophages and cytotoxic T lymphocytes in the glomeruli.

  • Neoliquiritin

    Neoliquiritin may possess ytotoxiciy and Tumor-specificity.